Friday, 10 January 2025

A Review on Nebivolol: Pharmacokinetic and Pharmacodynamics Approach | Chapter 7 | Pharmaceutical Research - Recent Advances and Trends Vol. 2

 

Nebivolol is one of the most recent β-blocking agents and it has vasodilating effects which may be useful in hypertensive patients with heart disease of ischemic (restriction in blood supply) origin or with erectile dysfunction. It is a third generation, long acting and highly selective β1 adrenergic receptor antagonist. It has a unique action that distinguishes it from other beta blockers. It increases the release of nitric oxide (NO) which produces vasodilatation via β3 receptor agonism. It improves endothelial function, which delays atherosclerosis. It improves arterial compliance and reduces peripheral vascular resistance and also reduces heart rate without improving maximal exercise tolerance. These effects are beneficial in hypertension and angina pectoris.

 

Author(s)details:-

 

Sahana G. N. (Associate Professor)
Department of Pharmacology, Hassan Institute of Medical Sciences, Hassan, India.

 

Sarala N. (Professor & HOD)
Department of Pharmacology, Sri Devaraj Urs Medical College, Tamaka, Kolar, India.

 

Kumar T. N. (Professor)
Department of Pharmacology Sri Narayana Institute of Medical Sciences, Ernakulum, Kerala, India.

 

Please See the book here :- https://doi.org/10.9734/bpi/prrat/v2/8270E

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